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Pharmacological characterization of novel allosteric enhancers of the A1 adenosine receptors
Varani, Katia; Romagnoli, Romeo; Vincenzi, Fabrizio; Targa, Martina; Preti, Delia; Baraldi, Pier Giovanni; Borea, Pier Andrea    
XXXIV Congresso Nazionale di Farmacologia, -
pp: ---, Anno: 2009

Synthesis and biological evaluation of new 8-heterocyclic xanthine derivative as highly potent and selective human A2B adenosine receptor antagonist
Baraldi, Pier Giovanni; Tabrizi, M. A.; Preti, Delia; Bovero, A.; Romagnoli, Romeo; Fruttarolo, Francesca; Zaid, N. A.; Moorman, A. R.; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 123-123, Anno: 2006

Recent developments in the field of A2B and A3 adenosine receptors antagonists
Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Zaid, N. A.; Moorman, A. R.; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 14-15, Anno: 2006

New 2-arylpyrazolo[4,3-c]quinoline derivates as potent and selective human A3 adenosine receptor antagonists
Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Fruttarolo, Francesca; Romagnoli, Romeo; Hussein, E. K.; Moormann, A. R.; Varani, Katia; Borea, Pier Andrea    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 325-325, Anno: 2006

Synthesis and biological characterization of [3H] 2-amino 4,5,6,7-tetrahydrobenzo(b)thiophen-3-yl-4-chloro phenyl methanone, the first radiolabeled adenosine A1 allosteric enhancer
Baraldi, Pier Giovanni; Pavani, Maria Giovanna; Iaconinoto, M. A.; Carrios, Y. Pelegrina M. D.; Cara, C. C.; Bowerman, S.; Varani, Katia; Moorman, A. R.; Romagnoli, Romeo    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 185-185, Anno: 2006

Synthesis and biological evaluation of allosteric A1 adenosine receptor modulators structurally related to 2-amino 4,5,6,7-tetrahydrobenzo(b) thiophen-3-yl-4-chloro phenyl methanone a potent compound useful to reduce neurophatic pain
Romagnoli, Romeo; Iaconinoto, M. A.; Carrion, M. D.; Cara, C. L.; Shryock, J. C.; Leung, E.; Moorman, A. R.; Gessi, Stefania; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 112-112, Anno: 2006

New pyrrolo [2,1-f] purine-2,4-dione and Imidazo[2,1-f]purine-2,4-dione derivates as potent and selective human A3 adenosine receptor antagonists
Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Zaid, N. A.; Moorman, A. R.; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea    
PURINERGIC SIGNALLING
Vol. 2, No. 1, pp: 270-270, Anno: 2006

New heterocyclic ligands for the adenosine receptors P1 and for the ATP receptors P2.
Baraldi, Pier Giovanni; AGHAZADEH TABRIZI, Mojgan; Preti, Delia; Bovero, Andrea; Romagnoli, Romeo; Fruttarolo, Francesca; Pavani, G.; Iaconinoto, M. A.; Varani, Katia; Borea, Pier Andrea    
-, -
pp: 63-63, Anno: 2005

Biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptors
Avitabile, Arianna; Baraldi, Pier Giovanni; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Leung, E.; Iannotta, Valeria; Merighi, Stefania; Gessi, Stefania; Varani, Katia; Pancaldi, Cecilia; Cattabriga, Elena; Borea, Pier Andrea    
-, -
pp: ---, Anno: 2003

Recent developments in the field of adenosine receptor ligands.
Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Pavani, M. G.; Avitabile, Arianna; Bovero, Andrea; Preti, Delia; Nuez Carretero, M. C.; Varani, Katia; Borea, Pier Andrea    
-, -
pp: 1-1, Anno: 2002

Recent developments in the field of adenosine receptor ligands
Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Cacciari, Barbara; Spalluto, G.; Romagnoli, Romeo; Pavani, M. G.; Nuez Carretero, M. C.; Varani, Katia; Borea, Pier Andrea    
Wiley, -
Vol. 56, No. 4, pp: 554-554, Anno: 2002

7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility.
Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea    
-, -
pp: ---, Anno: 2001

New potent and selective human adenosine A3 receptor antagonists.
Varani, Katia; Gessi, Stefania; Merighi, Stefania; Iannotta, Valeria; Leung, E.; Klotz, K. N.; Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Borea, Pier Andrea    
PHARMACOLOGICAL RESEARCH
Vol. 43, No. 1, pp: 17-17, Anno: 2001

New potent and selective human adenosine A3 receptor antagonists
Varani, Katia; Gessi, Stefania; Merighi, Stefania; Iannotta, Valeria; E., Leung; K. N., Klotz; Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Borea, Pier Andrea    
Società Italiana di Farmacologia, -
Vol. -, No. 1, pp: ---, Anno: 2001

7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility.
Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea    
-, -
pp: ---, Anno: 2001

Synthesis and molecular investigation of new pyrazolo[4,3-e]1,2,4,-triazolo[1,5-c]pyrimidine derivates as human A3 adenosine receptor antagonists.
Cacciari, Barbara; Moro, S.; Romagnoli, Romeo; Baraldi, Pier Giovanni; Gessi, Stefania; Pastorin, G.; Da Ros, T.; Varani, Katia; Borea, Pier Andrea; Spalluto, Giampiero    
-, -
pp: ---, Anno: 2001

Synthesis and molecular investigation of new pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivates as human A3 adenosine receptor antagonists.
Baraldi, Pier Giovanni; Cacciari, Barbara; Moro, S.; Romagnoli, Romeo; Gessi, Stefania; Pastorin, G.; De Ros, T.; Varani, Katia; Borea, Pier Andrea; Spalluto, Giampiero    
-, -
pp: ---, Anno: 2001

Pyrazolo[4,3-e]1,2,4-triazolo[1,5]pyrimidine derivates as irreversible antagonists at the human A3 adenosine receptor
Baraldi, Pier Giovanni; Cacciari, Barbara; Moro, S.; Romagnoli, Romeo; Xiao duo, J.; Jacobson, K.; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea; Spalluto, Giampiero    
International Union of Pure and Applied Chemistry, -
pp: ---, Anno: 2001

Pyrazolo [4,3-E]1,2,4-triazolo[1,5-c]pyrimidine derivates a new class of potent and selective human A3 adenosine receptor antagonists.
Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Klotz, K. N.; Leung, E.; Varani, Katia; Merighi, Stefania; Gessi, Stefania; Borea, Pier Andrea    
DRUG DEVELOPMENT RESEARCH
Vol. 50, No. 1, pp: 6-6, Anno: 2000

Pyrazolo-triazolo-pyrimidine derivates as adenosine receptor ligands: a search for A2B adenosine receptor antagonists.
Cacciari, Barbara; Spalluto, Giampiero; Baraldi, Pier Giovanni; Romagnoli, Romeo; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea    
-, -
pp: ---, Anno: 2000

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